1.1
Reagents:
Diisopropylethylamine
Catalysts:
Bis(dibenzylideneacetone)palladium
,
Tri-tert-butylphosphonium tetrafluoroborate
Solvents:
1,4-Dioxane
;
20 h, 100 °C
1.2
Reagents:
Sodium bicarbonate
,
Ammonium carbamate
Catalysts:
Bis(dibenzylideneacetone)palladium
,
(2R)-1-[(1R)-1-[Bis(1,1-dimethylethyl)phosphino]ethyl]-2-(diphenylphosphino)ferr…
Solvents:
1,4-Dioxane
;
20 h, 100 °C